SUMMARY; MD & MC; Modelling of counterions effects ...



 	Hi Netters,
 		This is the summary of my question about how to
 	model counterions in a DNA simulations ( polyelectrolytes
 	in general, but all the replies were DNA orientated ).
 	There was quite a lot of interest from people wanting to know
 	answers, and no clear concensus on 'How To', which must mean
 	a fruitful area of study.
 		From all these replies, and thinking about it myself,
 	I've formulated my own ideas along the lines of:
 		(1) It is well established that the DNA is only partially
 	neutralised in solution, both from ion condensation theory,
 	and from EXPERIMENT
 	( ie R. Podgornik et al, Biophys. J. 66 (1994) pp. 962-971
 	  which concludes that the DNA is only half neutralised, although
 	  this is for ordered DNA. )
 		(2) If we wish to model a section of partially neutralised
 	DNA, then it must only have a fraction of the counterions directly
 	site-bound to phosphates ( although QM work, I believe, predicts the
 	most electronegative areas to be the grooves and not the phosphates),
 	and the other counterions in the counterion atmosphere.
 		If we are using an explicit water box,
 	then we can either model with all the counterions in the box
 	( thus forcing the counterions from the distant atmosphere into
 	  the box )
 	or just exclude the counterions in the atmosphere and model a
 	negatively charged system, that is, apply a cutoff.
 		It seems like most people modelling DNA apply the
 	first method, forcing distant counterions to be local.
 		My OWN thoughts are that the second method seems more
 	natural, but not having done any 'charged'-DNA simulations I
 	cannot say anything about how stable it is. I would imagine that
 	the DNA would melt due to the repulsive -ve charges between the
 	chains ...
 		... now to the thoughts of others ...
 	( G. Ravishanker extensive reply was sent to the net previously,
 	  so it is not repeated here for bandwidth sake. )
 	Thanks for all the interest,
 				Kevin.
 -----------------------------------------------------------------------------
 From: "Virendra K. Saxena" <saxena { *at * } physics.purdue.edu>
        We did theoretical modeling of counterions around DNA using manning's
      ideas of "site-bound" and "area-bound" counterions, for
 the purpose of
      determining vibrational modes of DNA-counterion-water system. If you
      are interested in details please see: V. K. saxena and L. L. Van Zandt,
      Phys. Rev. A45, p7610-7620 (1992). If you get more information/discussion
      on this subject, please send me a copy. Thnaks,
          V. K. saxean
                Saxena
          saxena { *at * } physics.purdue.edu
 -----------------------------------------------------------------------------
 From: Tom Connor Bishop <bishop { *at * } lisboa.ks.uiuc.edu>
 kevin,
 i'm faced with the same DNA/couterion problem.
 please, let me know what others say.
 I'm modeling protein/DNA and found as
 expected that for only DNA in water, the
 DNA changed significantly
 from B-form.
 but the DNA with a significant amount of protein
 remained stable. the protein has + charge so i did
 not include counter ions in the dynamics. All said
 and done i have -24e on 18bp.
 For my system the protein binds in the
 major groove of the DNA, so groove widths
 are preserved more or less by the protein,
 which i think really helps, too.
 Do you know if there is a consensus as
 to whether or not the "deviations from B-form"
 that are found in simulations of DNA withOUT
 counter ions are "interpreted" as problems with MD
 for charged systems or as the real structural
 changes expected for DNA without ions.
 a reference on this would be great!
 thanks,
 tom
 -----------------------------------------------------------------------------
 From: Pieter Stouten <stoutepf { *at * } chemsci1.es.dupont.com>
 Hi Kevin,
 After having put the solute in a water box, I always calculate (using the
 program PROION that is part of the GROMOS distribution) the electrostatic
 potential on all water oxygen positions and replace the water molecule at
 the position with highest (positive or negative) potential with the
 appropriate ion. After placement of the counter ion, the ESP is
 recalculated and the next ion is placed. One continues until all positive
 and negative counter ions that one wants to use have been placed. This, of
 course is not the optimal solution for positioning more than one counter
 ion, but it has worked well for me so far.
 Cheers, Pieter.
 ** We have intermittent e-mail problems. If mail to me bounces back to you **
 ** please forward the bounced mail to stoutepf { *at * } lldmpc.dnet.dupont.com.
 **
 Pieter Stouten, Senior Research Scientist    ||
 Computer Aided Drug Design Group             ||
 The Du Pont Merck Pharmaceutical Company     ||    Adventures get spoiled
 P.O. Box 80353, Wilmington, DE 19880-0353    ||   by being reduced to data
 Phone: +1 (302) 695 3515                     ||             --
 Fax: +1 (302) 695 4324 (or 695 2813)         ||        Poul Anderson
 E-mail: stoutepf { *at * } chemsci1.es.dupont.com      ||
 Internet Shogi Server: kzinti                ||
 -----------------------------------------------------------------------------
 From: paul swartz <F0196903 { *at * } JAGUAR.CSC.WSU.EDU>
 Dear Mr. Bryson,
 	I have considered the same question that you put forth.  I do not
 know why full counter ion pairing is used though I have some ideas.  First,
 the first attempts in reducing the coulombic force due to explicit charges
 was done with a continuum approach in which all explicit charges were scaled
 by a constant factor.  Then the use of explicit counterions came along and
 the continuum approach was again used, all explicit charges were addressed.
 	Anothe factor is that most computational researchers interested in
 electrostatic forces and pot6ential fields ultimately want to apply
 Ewald sums in the propagation of their dynamics.  Ewald sums requires that the
 net charge of the system be zero.  It then requires that each charge have a
 counter charge though pairing is not required.  Additionally, most researchers
 seem to want to go toward the explicit treatment of physical effects and away
 from continuum approximations.
 Paul D. Swartz
 Washingto State University
 Pullman, WA 99163
 USA
 Email: F0196903 { *at * } jaguar.csc.wsu.edu
 Phone: 509-335-4083
 -----------------------------------------------------------------------------
 From: peter { *at * } vax.molecular-biophysics.oxford.ac.uk
 Dear Kevin,                                            7th July 1994
 Interesting thoughts about DNA counter-ions.   We hope to have a little
 paper in J.Mol.Graphics (Cruciani and Goodford) coming out about now.
 As a control we tried counter-ions at a range of distances from the
 phosphates, and found that it did not make too much difference to the Grid
 results in the minor groove.   I think this is because the electrostatic
 energy is a 1/r effect, and does not depend as critically on the distance
 as (for example) the Lennard-Jones energy which depends on 1/r**6.
 Of course, if you change the total number of counter-ions you will change
 the results dramatically.   In Grid, with a very negative Target like DNA;
 no counter-ions; and a negative Probe like carboxyl, the Probe will try
 to run away into the corners of the Grid cage.   I have therefore tended
 to study electrically neutral systems, not least because the real world
 is electrically neutral.
 Please keep me posted as other replies to your interesting question arrive.
 Best Regards.
 Peter Goodford.                                    peter { *at * }
 biop.oxford.ac.uk
 -----------------------------------------------------------------------------
 From: alex { *at * } mmiris.ab.umd.edu
 Kevin/Ravi,
    I have recently applied the new charmm all-hydrogen nucleic acid
 parameters to simulate a GCGCGCG and an ATATATA duplex in aqueous
 solution including approx. 0.9 M sodium and 0.5 M chloride yeilding
 a total charge 0.0 on the system.  Cutoffs were 12 A.  Periodic
 boundary conditions.  Without the use of any constraints stable
 structures were obtained for both systems during 500 ps simulations.
 In these calculations full charges were used.  The parameter paper has
 recently been submitted for publication and the results of the
 GCGCGCG and ATATATA simulations are in preparation.  The parameters
 themselves are currently available with the releases of charmm23 and
 charmm24.
 As I am primary author of the parameters consider this a biased
 opinion.
 Alex MacKerell, alex { *at * } mmiris.ab.umd.edu
 School of Pharmacy
 University of Maryland at Baltimore
 20 North Pine Street
 Baltimore, MD  21201
 410-706-7442
 -----------------------------------------------------------------------------