Second Swiss Course on Medicinal Chemistry



 Second Swiss Course on Medicinal Chemistry
 6-11 October 1996, Leysin, Switzerland
 organized by
 the Section of Medicinal Chemistry of the
 New Swiss Chemical Society
 SCOPE OF THE COURSE
 The course on medicinal chemistry offers to young scientists with a few
 years of experience in the pharmaceutical industry and interested Ph.D.
 students a broad overview of disciplines involved in modern preclinical drug
 research. The development of integrative abilities is a prerequisite to
 function in todays multidisciplinary drug discovery teams. The course is set
 up for synthetic organic chemists, as well as biologists and pharmacologists
 and those involved in drug design and the physicochemical characterization
 of biologically active compounds. Active participation by the participants
 in tutorials and the presentation of three case histories are important
 parts of the course.
 PROGRAMME AND LECTURERS
 What is medicinal chemistry?	Prof. B. Testa (Uni. Lausanne, CH)
 Molecular & Cell Biology
 What are the targets for the medicinal chemist	Dr. W. Schilling (Ciba, Basle
 - CH)
 Introduction to molecular biology 	Prof. T.H. Schwartz (Uni. Copenhagen, DK)
 Integration of molecular biology with medicinal chemistry	 Prof. T.H.
 Schwartz (Uni. Copenhagen, DK)
 Introduction to molecular immunology	Dr. J.-Y. Bonnefoy (Glaxo, Geneva - CH)
 Lead  Finding & Development
 Lead discovery	Dr. M. Sills (Ciba, Summit - USA)
 Introduction to combinatorial chemistry	Dr. E. Feder (Ciba, Basle- CH)
 Developing a lead	Dr. D. Roberts (Zeneca, Macclesfield - UK)
 Patents and regulatory apects	Dr. R. Ross (Sandoz, Basle - CH)
 Pharmacodynamics
 Principles of pharmacological assays	Prof. H. Möhler (Uni. Zürich, CH)
 Ion channels as drug targets	Prof. U. Quast (Uni. Tübingen, D)
 Phamacokinetics, Toxicology & Drug Delivery
 Introduction to pharmacokinetics	Prof. H. Spahn-Langguth (Uni. Halle, D)
 Introduction to drug metabolism	Prof. B. Testa (Uni. Lausanne, CH)
 Introduction to molecular toxicoloy	Prof. N.P.E. Vermeulen (Uni. Leiden, NL)
 Formulation and drug delivery	Prof. D. Crommelin (Uni. Utrecht, NL)
 Molecular Design & Lead Optimization
 Physicochemical concepts and drug absorption	Dr. H. van de Waterbeemd
 (Roche, Basle - CH)
 Molecular modeling	Prof. G. Folkers (ETH Zürich, CH)
 Computer-assisted lead optimization	Prof. H. Kubinyi (BASF, Ludwigshafen - D)
 Case Histories
 Development of aromatase inhibitors	Prof. A. Bhatnagar (Ciba, Basle - CH)
 The story of LESCOL	Dr. F. Kathawala (Sandoz, East Hanover - USA)
 Development of INVIRASE	Dr. J. Lawton (Roche, Welwyn - UK)
 ORGANIZATION
 Prof. Gerd Folkers (ETHZ, chairman), Dr. H. van de Waterbeemd (Roche,
 vice-chairman)
 Dr. W. Froestl (Ciba), Dr. R. Jakob-Roetne (Roche), Dr. D. Rognan (ETHZ),
 Prof. B. Testa (Uni. Lausanne), Dr. R. Wenger (Sandoz)
 WORLD WIDE WEB
 A description of the course including programme, location, accomodation
 facilities and registration form can be found at the following URL:
 http://www.pharma.ethz.ch/leysin
 PRACTICAL INFORMATIONS
 Location
 The course will be held at the Classic Hotel in Leysin, Switzerland. In the
 heart of the ?Alpes Vaudoises? and within easy reach of the towns of the
 Lake Geneva Region, Leysin is the perfect answer to the wishes and
 expectations of all those who love nature, winter and summer sports, walks,
 good food, the opportunity to meet interesting people, relaxation.
 Hotel
 The Classic is the largest hotel in Leysin, within the spirit of the resort.
 It offers a large array of single and double rooms, bars, restaurants,
 terrace, auditorium/cinema, gastronomic events.
 Registration fees
 The individual fee of Sfr 2500,- includes hotel accomodation with breakfast,
 course documentation, coffee breaks, lunches and dinner. Students pay a
 special price of only SFr 250,-  (please include justification to your
 registration)
 Registration
 The registration form should be returned before the end of April 1996. The
 course is limited to about 60 participants. Confirmation and payment
 instructions will be sent to all accepted participants. Late registrations
 after May 1st 1996 will require 10% additional fee.
 Arrival
 Sunday October 11, 1996 in the afternoon. Welcome drink at 6 p.m.
 Language
 The official language of the course is English.
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 REGISTRATION FORM
 Second Swiss Course on Medicinal Chemistry (6-11 October 1996, Leysin,
 Switzerland)
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 Please return this form to:
 Prof. Gerd Folkers, Dpt. of Pharmacy - ETH Wintherturerstrasse 190- CH-8057
 Zürich, Switzerland
 Tel. +41.1.257 60 60, Fax: +41.1.262 15 80, E-mail: folkers |-at-|
 pharma.ethz.ch
 Payments should be made to:
 Bankaccount 0061-867802-80-1 of Crédit Suisse  Claraplatz, CH-4005 Basel,
 Switzerland. (Ref: Swiss Med Chem)
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 Dr. Didier Rognan
 Department of Pharmacy - ETH
 Winterthurerstr.190, Room I17M50
 CH-8057 Zuerich
 phone:+41.1.257 60 63
 fax:  +41.1.262 15 80
 email: didier |-at-| pharma.ethz.ch
 www:  http://www.pharma.ethz.ch/~didier
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